Rauwolscine, tritiated on the methyl group. Rauwolscine acts as an antagonist at α2-adrenergic receptors.
Feature | Specification |
---|---|
Concentration | 1 mCi/ml |
Label Position | Specifically Labeled |
Molecular Weight | 354.4 |
Receptor | Adrenoceptors |
Rauwolscine, tritiated on the methyl group. Rauwolscine acts as an antagonist at α2-adrenergic receptors.
Rauwolscine acts as an α2-adrenergic receptor antagonist.
We offer both agonist and antagonist radioligands for autoradiographic visualization or performing saturation and competition assays to determine receptor expression levels (Bmax), dissociation constants (Kd), association and dissociation rates (kon and koff), and inhibitor constants (Ki) for a variety of receptors. We develop our radioligands to the highest specific activity possible and provide high purity resulting in low non-specific binding products. Each of our ultra-pure radioligands is fully characterized for pharmacological action and validated in receptor binding assays.
Radiolabeled ligands remain the most sensitive method for probing receptor binding biology; yielding unprecedented sensitivity gives results that technicians and scientists can trust. For over 50 years, Revvity has been a leading supplier of New England Nuclear (NEN) radiochemicals, liquid scintillation cocktails, vials and nuclear counting detection instruments.
References for NET722:
Concentration |
1 mCi/ml
|
---|---|
Molecular Weight |
354.4
|
Specific Activity |
>70 Ci/mmol (>2590 GBq/mmol)
|
CAS Number |
131-03-3
|
Application |
Drug Discovery & Development
|
---|---|
Brand |
NEN Radiochemicals
|
Buffer/Solvent |
Ethanol solution containing 0.25% ascorbic acid
|
Detection Modality |
Radiometric
|
Label Position |
Specifically Labeled
|
Molecular Formula |
C21H26N2O3
|
Packaging |
NENSure vial
|
Radioisotope |
3H
|
Receptor |
Adrenoceptors
|
Shipping Information |
Shipped in dry ice
|
Shipping Conditions |
Shipped in Dry Ice
|
Special Ordering Information |
This is a radioactive product - shipping address must have a license to receive radioactive materials.
|
Storage Conditions |
-80°C
|
Therapeutic Area |
Cardiovascular
|
Unit Size |
250 µCi
|
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